SCHEMBL8920848

SCHEMBL8920848

NC(=O)CN1C(=O)C(N)CC(c2ccccc2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.47
CCKBR P32239 12/20 0.44
SIGMAR1 Q99720 2/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541664 0.91 CCKBR (0.48) CYP2C19CCKBR
SCHEMBL9540219 0.91 CCKBR (0.47) CYP2C19CCKBR
SCHEMBL9540184 0.91 CYP2C19 (0.43) CYP2C19CCKBR
SCHEMBL9541670 0.88 CCKBR (0.51) CYP2C19CCKBRKMT2A
SCHEMBL9366810 0.88 CYP2C19 (0.47) CYP2C19CCKBRSIGMAR1RAB9AKMT2A
SCHEMBL9544115 0.86 CYP2C19 (0.46) CYP2C19RAB9A
SCHEMBL9544058 0.86 CCKBR (0.47) CYP2C19CCKBRSIGMAR1KMT2A
SCHEMBL9542926 0.86 CCKBR (0.49) CYP2C19CCKBRKMT2A
SCHEMBL8398546 0.86 CCKBR (0.48) CCKBR
SCHEMBL9542930 0.85 SLC6A2 (0.45) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
EP-0625145-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1994-11-23 EP disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed