SCHEMBL9541318

SCHEMBL9541318

O=C1NC(=O)C(N2C(=O)c3cccc4cccc(c34)C2=O)N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 1/20 0.46
ERCC1 P07992 1/20 0.46
FEN1 P39748 1/20 0.46
ERCC4 Q92889 1/20 0.46
PARP1 P09874 1/20 0.44
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TYMS P04818 1/20 0.42
HEXA P06865 3/20 0.41
HEXB P07686 3/20 0.41
TDP1 Q9NUW8 1/20 0.40
CES2 O00748 1/20 0.40
BCHE P06276 1/20 0.40
CES1 P23141 1/20 0.40
MCL1 Q07820 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11422629 0.85 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDHSD17B10TDP1
SCHEMBL20443756 0.78 DDB1 (0.55) ALDH1A1KDM4EHPGDNPSR1AKR1B1
SCHEMBL23409881 0.71 APP (0.39) ALDH1A1KDM4EHSD17B10MAPT
SCHEMBL24317510 0.69 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL2175176 0.69 CRBN (0.78) ALDH1A1TDP1MCL1CYP1A2
SCHEMBL862546 0.68 ERCC1 (0.63) CYP1B1ERCC1FEN1ERCC4PARP1
SCHEMBL9542756 0.66 DDB1 (0.38)
SCHEMBL27752410 0.66 ERCC1 (0.65) CYP1B1ERCC1FEN1ERCC4PARP1
SCHEMBL24317505 0.65 DDB1 (0.51) ALDH1A1HPGDMEN1KMT2ATDP1
SCHEMBL24453236 0.64 ERCC1 (0.63) CYP1B1ERCC1FEN1ERCC4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013092-A1 IMIDAZOLIDINEDIONE DERIVATIVES SARGES REINHARD (US) 1993-07-08 WO claimed
US-5011840-A Imidazolidinedione derivatives in diabetes treatment PFIZER INC. (US) 1991-04-30 US claimed
EP-0269355-B1 IMIDAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1991-04-10 EP claimed
EP-0269355-A1 Imidazolidinedione derivatives PFIZER INC. (US) 1988-06-01 EP claimed
WO-1993013092-A1 IMIDAZOLIDINEDIONE DERIVATIVES SARGES REINHARD (US) 1993-07-08 WO disclosed
WO-1993013092-A1 IMIDAZOLIDINEDIONE DERIVATIVES SARGES REINHARD (US) 1993-07-08 WO disclosed
US-5011840-A Imidazolidinedione derivatives in diabetes treatment PFIZER INC. (US) 1991-04-30 US disclosed
US-5011840-A Imidazolidinedione derivatives in diabetes treatment PFIZER INC. (US) 1991-04-30 US disclosed
EP-0269355-B1 IMIDAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1991-04-10 EP disclosed
EP-0269355-A1 Imidazolidinedione derivatives PFIZER INC. (US) 1988-06-01 EP disclosed