SCHEMBL9541502

SCHEMBL9541502

COc1ccc2[nH]c(=O)n(CCCCN3CCN(c4cccc(C(F)(F)F)c4)CC3)c2c1.O=c1[nH]c2ccccc2n1CCCN1CCN(c2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.71
ABCB11 O95342 1/20 0.71
ADRA2A P08913 1/20 0.71
ADORA3 P0DMS8 1/20 0.71
CHRM1 P11229 1/20 0.71
DRD1 P21728 1/20 0.71
TBXA2R P21731 1/20 0.71
SLC6A4 P31645 1/20 0.71
ADRA1A P35348 1/20 0.71
OPRM1 P35372 1/20 0.71
DRD3 P35462 1/20 0.71
KCNH2 Q12809 1/20 0.71
HTR7 P34969 11/20 0.60
ABCB1 P08183 2/20 0.53
DRD2 P14416 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
HTR6 P50406 1/20 0.52
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128738 0.96 HTR1A (0.66) HTR1AABCB11ADRA2AADORA3CHRM1
SCHEMBL7587470 0.91 HTR1A (0.74) HTR1AABCB11ADRA2AADORA3CHRM1
SCHEMBL8121534 0.90 HTR1A (0.88) HTR1AABCB11ADRA2AADORA3CHRM1
SCHEMBL8121051 0.90 HTR1A (0.88) HTR1AABCB11ADRA2AADORA3CHRM1
SCHEMBL8943053 0.89 HTR1A (0.86) HTR1AABCB11ADRA2AADORA3CHRM1
SCHEMBL8126688 0.87 HTR7 (0.74) HTR1AABCB11ADRA2AADORA3CHRM1
SCHEMBL6606413 0.85 HTR1A (0.74) HTR1AABCB11ADRA2AADORA3CHRM1
Flibanserin SCHEMBL30249132 0.84 HTR1A (1.00) HTR1AABCB11ADRA2AADORA3CHRM1
Flibanserin SCHEMBL29399513 0.84 HTR1A (1.00) HTR1AABCB11ADRA2AADORA3CHRM1
Flibanserin SCHEMBL247579 0.84 HTR1A (1.00) HTR1AABCB11ADRA2AADORA3CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003016-A1 BENZIMIDAZOLONE DERIVATIVES AS 5-HT1A AND 5-HT2 ANTAGONISTS BOEHRINGER INGELHEIM ITALIA S.P.A. (IT) 1993-02-18 WO claimed