SCHEMBL9542370

SCHEMBL9542370

NCCCC([C]=O)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.46
HRH1 P35367 1/20 0.46
MAOA P21397 2/20 0.42
MMP2 P08253 3/20 0.41
EPHX1 P07099 1/20 0.41
ALPI P09923 1/20 0.39
PKM P14618 1/20 0.39
PTGS1 P23219 1/20 0.39
XIAP P98170 1/20 0.39
SLC7A5 Q01650 1/20 0.39
TAAR1 Q96RJ0 3/20 0.38
SLC6A2 P23975 2/20 0.38
CYP2A6 P11509 2/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19812641 0.89 EPHX1 (0.43) HTR2AHRH1MAOAMMP2EPHX1
SCHEMBL7279390 0.84 SIGMAR1 (0.42) SLC6A3SIGMAR1SMN1; SMN2
SCHEMBL7300322 0.82 CNR2 (0.44) MMP2SIGMAR1SMN1; SMN2
SCHEMBL10349571 0.82 SIGMAR1 (0.44) MAOASIGMAR1
SCHEMBL5049235 0.81 EPHX1 (0.46) MAOAEPHX1ALPIPKMPTGS1
SCHEMBL5050487 0.81 EPHX1 (0.46) MAOAEPHX1ALPIPKMPTGS1
SCHEMBL19812666 0.81 EPHX1 (0.46) MAOAEPHX1ALPIPKMPTGS1
SCHEMBL7294571 0.81 CSNK1E (0.50) MMP2
SCHEMBL1697450 0.80 CYP1A2 (0.48) MAOAEPHX1ALPIPKMPTGS1
SCHEMBL7266826 0.79 MME (0.45) EPHX1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993000359-A1 MODIFIED PEPTIDES TRANSPORTABLE INTO THE CENTRAL NERVOUS SYSTEM THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-01-07 WO claimed
WO-1993000359-A1 MODIFIED PEPTIDES TRANSPORTABLE INTO THE CENTRAL NERVOUS SYSTEM THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-01-07 WO disclosed