SCHEMBL9542908

SCHEMBL9542908

CC(C)(C)OC(=O)N1c2ccccc2C[C@@H]1CC(=O)N[C@@H](CCc1ccccc1)C(=O)N1Cc2ccccc2C[C@@H]1CC(=O)O

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACE P12821 10/20 0.45
ABCB11 O95342 1/20 0.44
HDAC8 Q9BY41 1/20 0.40
PDE3A Q14432 1/20 0.40
PTPN1 P18031 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9544802 0.90 ACE (0.46) ACEABCB11PTPN1
SCHEMBL9544279 0.84 CTSK (0.52) ACEABCB11HDAC8
SCHEMBL9543839 0.83 ACE (0.43) ACE
SCHEMBL9544975 0.82 CTSK (0.51) ACE
SCHEMBL9544256 0.82 CTSK (0.51) ACE
SCHEMBL9542916 0.79 ACE (0.39) ACEABCB11
SCHEMBL9543218 0.78 CYP1A2 (0.44) ACE
SCHEMBL9542952 0.77 ELANE (0.40) ACE
SCHEMBL9542953 0.77 ELANE (0.40) ACE
SCHEMBL9544106 0.76 ELANE (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993020099-A2 CCK AND/OR GASTRIN RECEPTOR LIGANDS FERRING B.V. (NL) 1993-10-14 WO claimed
WO-1993020099-A2 CCK AND/OR GASTRIN RECEPTOR LIGANDS FERRING B.V. (NL) 1993-10-14 WO disclosed