SCHEMBL9543743

SCHEMBL9543743

CCCC(CN(C)S(=O)(=O)c1cccc2cnccc12)NS(=O)(=O)c1cccc2cnccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 3/20 0.49
PRKCG P05129 3/20 0.49
PRKCB P05771 3/20 0.49
PRKCA P17252 3/20 0.49
PRKCH P24723 3/20 0.49
PRKCI P41743 3/20 0.49
PRKCE Q02156 3/20 0.49
PRKCQ Q04759 3/20 0.49
PRKCZ Q05513 3/20 0.49
PRKCD Q05655 3/20 0.49
PRKD1 Q15139 3/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
NFKB1 P19838 2/20 0.49
GLA P06280 1/20 0.49
LMNA P02545 2/20 0.48
PMP22 Q01453 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PRKACA P17612 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542120 0.85 PRKD3 (0.53) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9541305 0.83 PRKCG (0.59) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL10754020 0.78 MELK (0.48) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL10983757 0.78 PRKD3 (0.56) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9541258 0.77 FLT3 (0.62) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL10985713 0.77 PRKD3 (0.60) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL9542795 0.76 PRKCG (0.68) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL11279652 0.75 PRKD3 (0.54) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL7430002 0.75 MELK (0.50) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL5130721 0.74 PRKCG (0.66) PRKD3PRKCGPRKCBPRKCAPRKCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013072-A1 5-ISOQUINOLINESULFONAMIDE DERIVATIVES AS PROTEIN KINASE INHIBITING AGENTS ITALFARMACO S.P.A. (IT) 1993-07-08 WO disclosed