SCHEMBL9545145

SCHEMBL9545145

O=C(O)c1c(F)c2c(F)c(F)ccc2[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
TDP1 Q9NUW8 2/20 0.44
DAO P14920 3/20 0.39
PARP1 P09874 2/20 0.36
GRIK1 P39086 1/20 0.35
GRIK2 Q13002 1/20 0.35
GRIK3 Q13003 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
GPR84 Q9NQS5 1/20 0.34
PADI4 Q9UM07 2/20 0.34
JAK2 O60674 1/20 0.33
THRB P10828 1/20 0.33
GPR35 Q9HC97 1/20 0.33
PDPK1 O15530 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
APEX1 P27695 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7041118 0.82 KDM4E (0.50) KDM4ETDP1DAOPARP1PADI4
SCHEMBL31171910 0.77 EIF4A3 (0.43) KDM4ETDP1DAOEGLN1GPR84
SCHEMBL15546942 0.77 PKM (0.39) KDM4EDAOEGLN1GPR84THRB
SCHEMBL476755 0.71 KDM4E (0.72) KDM4ETDP1DAOPARP1GPR35
SCHEMBL30388663 0.71 KDM4E (0.72) KDM4ETDP1DAOPARP1GPR35
SCHEMBL9389006 0.70 DAO (0.54) DAO
SCHEMBL31146049 0.70 PTGS2 (0.36) DAOPARP1GRIK1LMNAHPGD
SCHEMBL31145935 0.70 PTGS2 (0.36) DAOPARP1GRIK1LMNAHPGD
SCHEMBL31145855 0.70 PIM1 (0.44) KDM4EALDH1A1CYP2C19
SCHEMBL27353990 0.70 HDAC3 (0.39) DAOGPR84ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5092922-A None JP disclosed
JP-H0592922-A ANTIBACTERIAL AGENT BAYER AG 1993-04-16 JP disclosed
US-4952695-A Cyclopropyl-6,7,8-trifluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic acid, intermediate for antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1990-08-28 US disclosed
US-4556658-A 7-Amino-1-cyclopropyl-6,8-difluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acids and antibacterial agents containing these compounds BAYER AKTIENGESELLSCHAFT (DE) 1985-12-03 US disclosed
JP-H00592922-A 0001-01-01 JP disclosed