SCHEMBL9545566

SCHEMBL9545566

CN1C(=O)[C@@](NC(=O)Nc2cccc(CNc3nnn[nH]3)c2)(C2CCCCC2)N=Cc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 12/20 0.44
BACE1 P56817 4/20 0.35
BACE2 Q9Y5Z0 4/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
NPY1R P25929 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545585 0.90 CCKBR (0.40) CCKBRBACE1BACE2
SCHEMBL9545602 0.84 CCKBR (0.42) CCKBRBACE1BACE2
SCHEMBL9545572 0.83 CCKBR (0.42) CCKBRBACE1BACE2
SCHEMBL9545574 0.79 CCKBR (0.43) CCKBRBACE1BACE2
SCHEMBL9218194 0.76 CCKBR (0.35) CCKBRBACE1BACE2
SCHEMBL9213794 0.76 BACE1 (0.35) CCKBRBACE1BACE2
SCHEMBL9701161 0.74 CCKBR (0.55) CCKBRBACE1BACE2
SCHEMBL9702299 0.74 CCKBR (0.55) CCKBRBACE1BACE2
SCHEMBL9699964 0.74 CCKBR (0.45) CCKBRBACE1BACE2SMN1; SMN2NPY1R
SCHEMBL9301937 0.74 CCKBR (0.55) CCKBRBACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993019052-A1 3-UREIDO SUBSTITUTED BENZODIAZEPIN-2-ONES HAVING CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTIC ACTIVITY AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-09-30 WO claimed
WO-1993019052-A1 3-UREIDO SUBSTITUTED BENZODIAZEPIN-2-ONES HAVING CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTIC ACTIVITY AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-09-30 WO disclosed