SCHEMBL9545602

SCHEMBL9545602

Cc1ccc(NC(=O)N[C@]2(C3CCCCC3)N=Cc3ccccc3N(C)C2=O)cc1Nc1nnn[nH]1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 12/20 0.42
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KCNJ6 P48051 1/20 0.31
KCNJ5 P48544 1/20 0.31
KCNJ3 P48549 1/20 0.31
LDLR P01130 1/20 0.31
APP P05067 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
MAPK14 Q16539 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545585 0.90 CCKBR (0.40) CCKBRBACE1BACE2
SCHEMBL9545574 0.84 CCKBR (0.43) CCKBRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9545566 0.84 CCKBR (0.44) CCKBRBACE1BACE2
SCHEMBL9545572 0.80 CCKBR (0.42) CCKBRBACE1BACE2
SCHEMBL9301948 0.78 CCKBR (0.41) CCKBRALDH1A1NPC1RAB9ALDLR
SCHEMBL9303570 0.75 CCKBR (0.45) CCKBRALDH1A1MAPK14MAPT
SCHEMBL9218194 0.73 CCKBR (0.35) CCKBRAPPCTSDBACE1BACE2
SCHEMBL9301587 0.72 CCKBR (0.57) CCKBRNPC1RAB9ABACE1BACE2
SCHEMBL14425315 0.72 CCKBR (0.77) CCKBR
SCHEMBL9545600 0.72 CCKBR (0.77) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993019052-A1 3-UREIDO SUBSTITUTED BENZODIAZEPIN-2-ONES HAVING CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTIC ACTIVITY AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-09-30 WO claimed
WO-1993019052-A1 3-UREIDO SUBSTITUTED BENZODIAZEPIN-2-ONES HAVING CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTIC ACTIVITY AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-09-30 WO disclosed