SCHEMBL9546857

SCHEMBL9546857

CC1C[C@@]2(C)[C@@H](CC[C@H]3[C@@H]4CCC[C@@]4(C)CC[C@@H]32)NC1=O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
NR1I3 Q14994 1/20 0.43
MBOAT4 Q96T53 3/20 0.41
GRIN1 Q05586 3/20 0.40
GRIN2B Q13224 3/20 0.40
CYP19A1 P11511 3/20 0.40
SRD5A1 P18405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9110720 0.86 NR1I3 (0.48) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL15549709 0.86 NR1I3 (0.48) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL8712727 0.84 CDK5 (0.41) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL7609110 0.83 GRIN1 (0.45) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL9547062 0.83 GRIN1 (0.45) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL9185884 0.82 CDK5 (0.42) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL8710575 0.82 GRIN1 (0.43) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL8707760 0.82 GRIN1 (0.42) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL8019796 0.80 GRIN1 (0.43) CDK5CDK5R1NR1I3MBOAT4GRIN1
SCHEMBL8710564 0.79 MBOAT4 (0.38) CDK5CDK5R1NR1I3MBOAT4GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993023039-A1 SUBSTITUTED 4-AZA-5A-ANDROSTAN-ONES AS 5A-REDUCTASE INHIBITORS MERCK & CO., INC. (US) 1993-11-25 WO disclosed