SCHEMBL9547703

SCHEMBL9547703

CCC(Cc1cnc2nc(N)nc(N)c2n1)(C(=O)OC)c1ccc(C(=O)OC)s1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
ATM Q13315 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NOS1 P29475 1/20 0.42
DHFR P00374 6/20 0.41
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9547730 0.84 DHFR (0.44) NOS1DHFRCA1CA2
SCHEMBL9547681 0.82 DHFR (0.45) NOS1DHFRCA1CA2
SCHEMBL15055178 0.75 DHFR (0.45) DHFR
SCHEMBL9313953 0.74 DHFR (0.43) DHFR
SCHEMBL9547710 0.70 DHFR (0.48) NOS1DHFRCA1CA2
SCHEMBL9067320 0.67 DHFR (0.47) DHFRCA1CA2
SCHEMBL9541999 0.67 DHFR (0.66) DHFR
SCHEMBL16980950 0.67 NOS1 (0.53) NOS1DHFR
SCHEMBL9542041 0.66 DHFR (0.52) DHFR
SCHEMBL20780857 0.66 NOS1 (0.67) NOS1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993022315-A1 HETEROAROYL-10-DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1993-11-11 WO disclosed