SCHEMBL9550010

SCHEMBL9550010

CCN1CCCC1CNC(=O)c1c(OC)c(N)cc(Br)c1OC

nearest known ligand 0.85

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.80
DRD4 P21917 2/20 0.70
DRD3 P35462 2/20 0.70
MEN1 O00255 1/20 0.70
HTR1A P08908 1/20 0.70
ADRA2A P08913 1/20 0.70
CYP2D6 P10635 1/20 0.70
ADRA2C P18825 1/20 0.70
CYP2C19 P33261 1/20 0.70
ADRA1A P35348 1/20 0.70
HTR2B P41595 1/20 0.70
KMT2A Q03164 1/20 0.70
KCNH2 Q12809 1/20 0.70
HIF1A Q16665 1/20 0.70
SIGMAR1 Q99720 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9549997 1.00 DRD2 (0.80) DRD2DRD4DRD3MEN1HTR1A
SCHEMBL11163460 0.93 DRD2 (0.88) DRD2DRD4DRD3MEN1HTR1A
SCHEMBL9550072 0.92 DRD2 (0.80) DRD2DRD4DRD3
SCHEMBL9550077 0.92 DRD2 (0.80) DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL10691937 0.92 DRD2 (0.86) DRD2DRD4DRD3MEN1HTR1A
SCHEMBL9549931 0.89 DRD2 (1.00) DRD2
SCHEMBL9550067 0.89 DRD2 (0.85) DRD2DRD4DRD3MEN1HTR1A
SCHEMBL9549949 0.89 DRD2 (1.00) DRD2
SCHEMBL9550074 0.89 DRD2 (0.85) DRD2DRD4DRD3MEN1HTR1A
SCHEMBL11168904 0.88 DRD2 (0.80) DRD2DRD4DRD3MEN1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5240957-A Dopaminergic agent ASTRA LAKEMEDEL AKTEIBOLAG (SE) 1993-08-31 US disclosed
EP-0156776-A1 Derivatives of N-(2-pyrrolidinylmethyl)-benzamide, process for their preparation, intermediates and a pharmaceutical preparation Astra Läkemedel Aktiebolag (SE) 1985-10-02 EP disclosed