SCHEMBL9550722

SCHEMBL9550722

CCC(=O)CCSc1cc(-c2ccccc2)c(O)c(-c2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.42
PTPN6 P29350 2/20 0.42
PTPN2 P17706 1/20 0.42
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 4/20 0.37
HNF4A P41235 1/20 0.37
IAPP P10997 2/20 0.37
BACE1 P56817 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9551140 0.85 AKR1C3 (0.45) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9813051 0.85 PTPN1 (0.44) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9550710 0.85 ALDH1A1 (0.49) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9550715 0.82 PTPN1 (0.41) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9550720 0.82 BACE1 (0.42) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9551123 0.81 PTPN1 (0.36) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9550711 0.80 ALDH1A1 (0.47) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9813187 0.80 AKR1C3 (0.43) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL199038 0.79 ALDH1A1 (0.43) PTPN1PTPN6PTPN2AKR1C3AKR1C2
SCHEMBL9838242 0.77 TDP1 (0.44) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229421-A Antiallergens, antiinflammatory agents G. D. SEARLE & CO. (US) 1993-07-20 US disclosed
EP-0339688-B1 HYDROXYPHENYLTHIOALKYLKETONES G.D. Searle & Co. (US) 1993-03-10 EP disclosed
US-4857558-A ANTIINFLAMMATORY AGENTS AND-OR ANTIALLERGENS G. D. SEARLE & CO. (US) 1989-08-15 US disclosed