SCHEMBL9550720

SCHEMBL9550720

COC(=O)CCSc1cc(-c2ccccc2)c(O)c(-c2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.42
PTGS1 P23219 1/20 0.42
ATM Q13315 1/20 0.42
PTPN1 P18031 5/20 0.41
PTPN2 P17706 1/20 0.41
PTPN6 P29350 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.40
APP P05067 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
LTB4R Q15722 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 1/20 0.40
PRNP P04156 1/20 0.40
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9813051 0.84 PTPN1 (0.44) BACE1PTPN1PTPN2PTPN6ALDH1A1
SCHEMBL9550710 0.84 ALDH1A1 (0.49) PTPN1PTPN2PTPN6ALDH1A1CYP1A2
SCHEMBL9550722 0.82 PTPN1 (0.42) BACE1PTPN1PTPN2PTPN6ALDH1A1
SCHEMBL9550715 0.81 PTPN1 (0.41) BACE1PTPN1PTPN2PTPN6ALDH1A1
SCHEMBL19274345 0.81 LTB4R (0.45) ATMALDH1A1LMNAAPPCYP1A2
SCHEMBL28897181 0.80 CYP1A2 (0.59) ATMALDH1A1LMNACYP1A2CYP3A4
SCHEMBL9550711 0.79 ALDH1A1 (0.47) BACE1PTPN1PTPN2PTPN6ALDH1A1
SCHEMBL21016682 0.77 LTB4R (0.43) ATMPTPN1ALDH1A1LMNACYP1A2
SCHEMBL9510615 0.77 SMN1; SMN2 (0.53) ALDH1A1LMNAL3MBTL1
SCHEMBL9838242 0.76 TDP1 (0.44) ALDH1A1LMNACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229421-A Antiallergens, antiinflammatory agents G. D. SEARLE & CO. (US) 1993-07-20 US disclosed
US-5208262-A Administering 4-hydroxythiophenol derivatives G. D. SEARLE & CO. (US) 1993-05-04 US disclosed
EP-0339688-B1 HYDROXYPHENYLTHIOALKYLKETONES G.D. Searle & Co. (US) 1993-03-10 EP disclosed
US-5047593-A Antiinflammatory And Antiallergy Agents G. D. SEARLE & CO. (US) 1991-09-10 US disclosed
EP-0339688-A1 Hydroxyphenylthioalkylketones G.D. Searle & Co. (US) 1989-11-02 EP disclosed
US-4857558-A ANTIINFLAMMATORY AGENTS AND-OR ANTIALLERGENS G. D. SEARLE & CO. (US) 1989-08-15 US disclosed
EP-0218782-A1 Lipoxygenase-inhibiting composition and hydroxyphenylthioalkylcarbonyl compounds G.D. Searle & Co. (US) 1987-04-22 EP disclosed