SCHEMBL9550801

SCHEMBL9550801

OCCCSc1cc(-c2ccccc2)c(O)c(-c2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.41
PTPN6 P29350 2/20 0.41
PTPN2 P17706 1/20 0.41
BACE1 P56817 3/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.39
BCL2L1 Q07817 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
CA2 P00918 1/20 0.39
MAPK1 P28482 1/20 0.38
ALOX5 P09917 1/20 0.36
HNF4A P41235 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9554837 0.87 BACE1 (0.47) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL199038 0.87 ALDH1A1 (0.43) PTPN1PTPN6PTPN2BACE1ALDH1A1
SCHEMBL202457 0.84 SOAT1 (0.42) HDAC2
SCHEMBL9550711 0.82 ALDH1A1 (0.47) PTPN1PTPN6PTPN2BACE1ALDH1A1
SCHEMBL9555047 0.81 CA2 (0.47) BACE1ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL9550710 0.80 ALDH1A1 (0.49) PTPN1PTPN6PTPN2ALDH1A1AKR1C3
SCHEMBL9551146 0.78 BACE1 (0.39) PTPN1PTPN6PTPN2BACE1ALDH1A1
SCHEMBL9813051 0.78 PTPN1 (0.44) PTPN1PTPN6PTPN2BACE1ALDH1A1
SCHEMBL9551121 0.77 BACE1 (0.34) PTPN1PTPN6PTPN2BACE1ALDH1A1
SCHEMBL95857 0.77 ALDH1A1 (0.64) ALDH1A1CA2MAPK1HDAC4HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229421-A Antiallergens, antiinflammatory agents G. D. SEARLE & CO. (US) 1993-07-20 US disclosed
US-5208262-A Administering 4-hydroxythiophenol derivatives G. D. SEARLE & CO. (US) 1993-05-04 US disclosed
US-5047593-A Antiinflammatory And Antiallergy Agents G. D. SEARLE & CO. (US) 1991-09-10 US disclosed
EP-0218782-B1 LIPOXYGENASE-INHIBITING COMPOSITION AND HYDROXYPHENYLTHIOALKYLCARBONYL COMPOUNDS G.D. Searle & Co. (US) 1990-05-16 EP disclosed
US-4857558-A ANTIINFLAMMATORY AGENTS AND-OR ANTIALLERGENS G. D. SEARLE & CO. (US) 1989-08-15 US disclosed
EP-0218782-A1 Lipoxygenase-inhibiting composition and hydroxyphenylthioalkylcarbonyl compounds G.D. Searle & Co. (US) 1987-04-22 EP disclosed