SCHEMBL9553453

SCHEMBL9553453

c1ccc(-c2nc(Cc3ccc(-c4ccccc4-c4nnn[nH]4)cc3)n(C3CCCCC3)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
TRPV1 Q8NER1 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC33A1 O00400 2/20 0.35
KCNJ6 P48051 4/20 0.35
KCNJ5 P48544 4/20 0.35
KCNJ3 P48549 4/20 0.35
S1PR1 P21453 2/20 0.35
AGTR1 P30556 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTSK P43235 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9553197 0.89 SLC33A1 (0.35) ALDH1A1TRPV1SLC33A1KCNJ6KCNJ5
SCHEMBL9552746 0.88 SLC33A1 (0.36) ALDH1A1TRPV1SLC33A1KCNJ6KCNJ5
SCHEMBL9552478 0.88 SLC33A1 (0.36) ALDH1A1TRPV1SLC33A1KCNJ6KCNJ5
SCHEMBL9553327 0.87 SLC33A1 (0.35) ALDH1A1TRPV1SLC33A1KCNJ6KCNJ5
SCHEMBL9553553 0.86 AGTR1 (0.37) TRPV1SLC33A1KCNJ6KCNJ5KCNJ3
SCHEMBL9552076 0.86 SLC33A1 (0.35) ALDH1A1TRPV1SLC33A1KCNJ6KCNJ5
SCHEMBL9552812 0.86 SLC33A1 (0.38) TRPV1SLC33A1KCNJ6KCNJ5KCNJ3
SCHEMBL9552356 0.86 RIPK1 (0.37) ALDH1A1TRPV1SLC33A1KCNJ6KCNJ5
SCHEMBL9552169 0.85 AGTR1 (0.35) SLC33A1S1PR1AGTR1
SCHEMBL9553055 0.85 SLC33A1 (0.36) ALDH1A1TRPV1MEN1KMT2ASLC33A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229406-A Treatment of glaucoma G. D. SEARLE & CO. (US) 1993-07-20 US disclosed
US-5140036-A Hypotensive agents; congestive heart failure; angiotensin antagonists G. D. SEARLE & CO. (US) 1992-08-18 US disclosed
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO disclosed