SCHEMBL9554306

SCHEMBL9554306

COC(=O)[C@H](Cc1ccccc1)NC(=O)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.60
ALDH1A1 P00352 2/20 0.59
THRB P10828 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
HSD17B10 Q99714 1/20 0.59
POLB P06746 1/20 0.58
LMNA P02545 1/20 0.55
GLA P06280 1/20 0.55
PTGES O14684 2/20 0.54
PSEN1 P49768 2/20 0.54
PSEN2 P49810 2/20 0.54
APH1B Q8WW43 2/20 0.54
NCSTN Q92542 2/20 0.54
APH1A Q96BI3 2/20 0.54
PSENEN Q9NZ42 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
GAA P10253 1/20 0.53
RAB9A P51151 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9554565 0.85 PTPN1 (0.61) ALDH1A1PTGESL3MBTL1
SCHEMBL22634292 0.84 ATM (0.55) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL22634288 0.84 ATM (0.55) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL7806984 0.80 ATM (0.68) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL1884230 0.80 ATM (0.68) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL1879654 0.80 ATM (0.68) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL803579 0.80 ATM (0.68) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL6295802 0.80 ATM (0.68) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL11015260 0.80 ATM (0.60) ATMALDH1A1THRBCYP2C9CYP2C19
SCHEMBL22647465 0.79 ATM (0.50) ATMALDH1A1THRBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5250517-A Hypotensive and cardiotonic agents; cardiac insufficiency HOFFMANN-LA ROCHE INC. (US) 1993-10-05 US disclosed
EP-0386611-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1990-09-12 EP disclosed
EP-0310918-A2 Peptide-like amino-acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-04-12 EP disclosed