SCHEMBL9559129

SCHEMBL9559129

CCCCCN(CCOC(C)=O)C(=O)C(CCC(=O)OCc1ccccc1)CS(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 5/20 0.45
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MMP1 P03956 1/20 0.35
MMP7 P09237 1/20 0.35
ACE P12821 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
CTRC Q99895 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9558893 0.90 CCKBR (0.47) CCKBRALDH1A1HPGDGAACA12
SCHEMBL9559037 0.88 GAA (0.46) CCKBRLMNAALDH1A1HPGDMEN1
SCHEMBL9558985 0.84 CCKBR (0.46) CCKBRALDH1A1HPGDMEN1KMT2A
SCHEMBL9558855 0.81 GAA (0.51) CCKBRLMNAALDH1A1HPGDMEN1
SCHEMBL9558960 0.81 CCKBR (0.46) CCKBRALDH1A1HPGDGAACA12
SCHEMBL9558862 0.80 CCKBR (0.51) CCKBRALDH1A1HPGDKDM4EMMP1
Water SCHEMBL9559012 0.79 CCKBR (0.50) CCKBRALDH1A1HPGDKDM4EMMP1
SCHEMBL9559024 0.79 CCKBR (0.46) CCKBRALDH1A1HPGDGAACA12
SCHEMBL9559135 0.78 GAA (0.49) CCKBRALDH1A1HPGDGAACA12
SCHEMBL9559158 0.78 GAA (0.48) CCKBRLMNAALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3197453-A None JP disclosed
US-5177069-A Cholecystokinin inhibitor, pancreatic antisecretory agent KISSEI PHARMACEUTICAL CO., LTD. (JP) 1993-01-05 US disclosed
JP-H03197453-A NAPHTHYLSULFONYLALKYLCARBOXYLIC ACID DERIVATIVE KISSEI PHARMACEUT CO LTD 1991-08-28 JP disclosed
EP-0433064-A1 Naphthylsulfonylalkanoic acid compounds Kissei Pharmaceutical Co., Ltd. (JP) 1991-06-19 EP disclosed