SCHEMBL9560118

SCHEMBL9560118

Cc1ccc(C(=S)C(C)N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
LMNA P02545 2/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
CTSL P07711 3/20 0.41
CTSB P07858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 3/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
PKM P14618 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1713136 0.81 ALDH1A1 (0.44) ALDH1A1LMNACES2CES1CTSL
SCHEMBL28879932 0.79 ADRA2C (0.46) ALDH1A1LMNAPKMATMMAOA
SCHEMBL7778314 0.77 ALDH1A1 (0.41) ALDH1A1LMNACES2CES1CTSL
SCHEMBL8995282 0.77 ALDH1A1 (0.41) ALDH1A1LMNACES2CES1CTSL
SCHEMBL9559836 0.75 PARP1 (0.50) ALDH1A1CTSLSMN1; SMN2HDAC8HDAC6
SCHEMBL11171647 0.74 ALDH1A1 (0.42) ALDH1A1LMNACES2CES1CTSL
SCHEMBL16694617 0.73 ALDH1A1 (0.52) ALDH1A1LMNACES2CES1SMN1; SMN2
SCHEMBL2631353 0.73 ALDH1A1 (0.52) ALDH1A1LMNACES2CES1SMN1; SMN2
SCHEMBL28228323 0.73 ALDH1A1 (0.52) ALDH1A1LMNACES2CES1SMN1; SMN2
SCHEMBL11186390 0.71 ALDH1A1 (0.39) ALDH1A1LMNACES2CES1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325247-B1 CAMPTOTHECIN DERIVATIVES AND PROCESS FOR PREPARING SAME KABUSHIKI KAISHA YAKULT HONSHA (JP) 1993-05-19 EP disclosed
US-5061800-A ANTITUMOR AGENTS KABUSHIKI KAISHA YAKULT HONSHA (JP) 1991-10-29 US disclosed
EP-0325247-A1 Camptothecin derivatives and process for preparing same KABUSHIKI KAISHA YAKULT HONSHA (JP) 1989-07-26 EP disclosed