SCHEMBL9564183

SCHEMBL9564183

CCC(c1ccc(C(=O)OC(C)(C)C)cc1)c1c[nH]c2nc(N)nc(O)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
DHFR P00374 2/20 0.34
TYMS P04818 2/20 0.34
ABCG2 Q9UNQ0 1/20 0.33
CHUK O15111 1/20 0.32
SLC7A5 Q01650 1/20 0.32
STAT3 P40763 2/20 0.31
SMO Q99835 1/20 0.31
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
GLA P06280 1/20 0.30
MAPK1 P28482 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564211 0.89 CA12 (0.34) CA12CA1CA2CA9CA14
SCHEMBL9564231 0.88 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL9564178 0.84 CA12 (0.34) CA12CA1CA2CA9CA14
SCHEMBL9564205 0.78 TYMS (0.43) DHFRTYMS
SCHEMBL9564203 0.76 DHFR (0.47) DHFRTYMSL3MBTL1
SCHEMBL9564145 0.74 DHFR (0.57) DHFRTYMS
SCHEMBL8997200 0.73 NAMPT (0.42) DHFRTYMS
SCHEMBL9564151 0.71 DHFR (0.49) DHFRTYMS
SCHEMBL9564180 0.71 DHFR (0.46) DHFRTYMSL3MBTL1
SCHEMBL9564181 0.71 DHFR (0.46) DHFRTYMSL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed