SCHEMBL9564211

SCHEMBL9564211

CC(C)(C)OC(=O)c1ccc(C(C[N+](=O)[O-])c2c[nH]c3nc(N)nc(O)c23)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
UBE2B P63146 1/20 0.32
DHFR P00374 1/20 0.31
TYMS P04818 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
NR1H4 Q96RI1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564183 0.89 CA12 (0.35) CA12CA1CA2CA9CA14
SCHEMBL9564231 0.83 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL9564178 0.80 CA12 (0.34) CA12CA1CA2CA9CA14
SCHEMBL9564168 0.78 DHFR (0.54) CA1CA2DHFRTYMS
SCHEMBL9564214 0.77 DHFR (0.43) DHFRTYMS
SCHEMBL9564218 0.77 DHFR (0.43) DHFRTYMS
SCHEMBL9564205 0.74 TYMS (0.43) DHFRTYMS
SCHEMBL9564143 0.69 TYMS (0.48) CA1CA2DHFRTYMS
SCHEMBL8997200 0.69 NAMPT (0.42) DHFRTYMS
SCHEMBL9564160 0.67 DHFR (0.58) CA1CA2DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed