SCHEMBL9564232

SCHEMBL9564232

Cc1nc(O)c2c(Cc3cnc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s3)c[nH]c2n1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 5/20 0.45
SLC19A1 P41440 5/20 0.45
SLC46A1 Q96NT5 5/20 0.45
TYMS P04818 8/20 0.45
DHFR P00374 4/20 0.45
GART P22102 3/20 0.44
FOLR2 P14207 1/20 0.41
ATIC P31939 1/20 0.41
SHMT1 P34896 1/20 0.41
FRK P42685 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564257 0.89 DHFR (0.51) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9221148 0.89 FOLR1 (0.49) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9228438 0.89 FOLR1 (0.49) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9564301 0.86 FOLR1 (0.59) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9221160 0.82 FOLR1 (0.44) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9564228 0.81 DHFR (0.67) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9439922 0.80 FOLR1 (0.57) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9228451 0.79 FOLR1 (0.42) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9228529 0.79 DHFR (0.53) FOLR1SLC19A1SLC46A1TYMSDHFR
SCHEMBL9226502 0.79 DHFR (0.53) FOLR1SLC19A1SLC46A1TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed