SCHEMBL9564301

SCHEMBL9564301

Cc1nc(O)c2c(Cc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s3)c[nH]c2n1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 11/20 0.59
SLC46A1 Q96NT5 8/20 0.59
SLC19A1 P41440 6/20 0.59
GART P22102 7/20 0.57
DHFR P00374 4/20 0.49
TYMS P04818 4/20 0.49
FOLR2 P14207 4/20 0.45
ATIC P31939 3/20 0.45
SHMT1 P34896 1/20 0.44
FRK P42685 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564163 0.90 FOLR1 (0.62) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9227773 0.89 FOLR1 (0.66) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9223823 0.89 FOLR1 (0.66) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564164 0.86 FOLR1 (0.53) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564232 0.86 FOLR1 (0.45) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564228 0.83 DHFR (0.67) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439839 0.82 FOLR1 (0.74) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564303 0.81 FOLR1 (0.48) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564236 0.81 FOLR1 (0.46) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564256 0.81 FOLR1 (0.49) FOLR1SLC46A1SLC19A1GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549291-A1 Thymidylate synthase inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed