SCHEMBL9564771

SCHEMBL9564771

c1ncc2nc(NC3CCNCC3)n(Cc3cscn3)c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN9A Q15858 2/20 0.35
SOS1 Q07889 1/20 0.35
CYP1A2 P05177 4/20 0.33
USP2 O75604 3/20 0.33
ALDH1A1 P00352 3/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALOX15 P16050 1/20 0.33
HIF1A Q16665 1/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
CDC42BPB Q9Y5S2 1/20 0.32
MAPK8 P45983 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564899 0.83 KCNH2 (0.40) NR4A2KCNH2SOS1CYP1A2USP2
SCHEMBL9564782 0.82 KCNH2 (0.45) NR4A2KCNH2SOS1CYP1A2USP2
SCHEMBL9564948 0.80 ALDH1A1 (0.42) ALDH1A1HSD17B10MAPK8CDK2TSHR
Bromide SCHEMBL9564796 0.79 NR4A2 (0.54) NR4A2KCNH2SOS1CYP1A2USP2
SCHEMBL9564960 0.79 CYP1A2 (0.43) NR4A2KCNH2CYP1A2USP2ALDH1A1
SCHEMBL9564845 0.78 KCNH2 (0.64) NR4A2KCNH2SOS1CYP1A2USP2
Hydrochloric Acid SCHEMBL9564856 0.78 KCNH2 (0.63) NR4A2KCNH2SOS1CYP1A2USP2
Bromide SCHEMBL9698211 0.78 KCNH2 (0.60) NR4A2KCNH2SOS1CYP1A2USP2
Bromide SCHEMBL9699552 0.78 KCNH2 (0.60) NR4A2KCNH2SOS1CYP1A2USP2
Bromide SCHEMBL9630147 0.77 NR4A2 (0.39) NR4A2KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed