SCHEMBL9565313

SCHEMBL9565313

O=c1[nH]cc(-c2cccnc2)nc1CC1CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.46
AURKA O14965 1/20 0.44
TTK P33981 1/20 0.44
AURKB Q96GD4 1/20 0.44
INCENP Q9NQS7 1/20 0.44
MAPK1 P28482 2/20 0.39
VCP P55072 1/20 0.38
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
METAP2 P50579 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
CYP19A1 P11511 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
HPGD P15428 1/20 0.36
MAPT P10636 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
RIPK3 Q9Y572 1/20 0.36
CYP3A4 P08684 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435148 0.77 PDGFRB (0.49) PDGFRBAURKATTKAURKBINCENP
SCHEMBL7430163 0.77 CYP11B1 (0.47) PDGFRBAURKATTKAURKBINCENP
SCHEMBL9565318 0.77 PDGFRB (0.48) PDGFRBAURKATTKAURKBINCENP
SCHEMBL9565316 0.75 CYP2A6 (0.43) MAPK1VCPCYP19A1CYP3A4CYP2A6
SCHEMBL9565370 0.74 PDGFRB (0.46) PDGFRBAURKATTKAURKBINCENP
SCHEMBL9565358 0.72 MAPK1 (0.41) MAPK1VCPCYP3A4CYP2A6PDE5A
SCHEMBL7434051 0.70 PDGFRB (0.52) PDGFRBAURKATTKAURKBINCENP
SCHEMBL23124200 0.69 MAPK1 (0.45) PDGFRBMAPK1PARP10PARP11METAP2
SCHEMBL7495544 0.68 PDGFRB (0.48) PDGFRBAURKATTKAURKBINCENP
SCHEMBL1435835 0.67 CYP2A6 (0.54) PDGFRBMAPK1PARP10PARP11METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543245-A1 Renin inhibiting amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed