SCHEMBL7435148

SCHEMBL7435148

CC(C)Cc1nc(-c2cccnc2)c[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.49
AURKA O14965 1/20 0.45
TTK P33981 1/20 0.45
AURKB Q96GD4 1/20 0.45
INCENP Q9NQS7 1/20 0.45
CYP2A6 P11509 2/20 0.40
MAPK1 P28482 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2E1 P05181 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM5B Q9UGL1 1/20 0.39
PIM1 P11309 1/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
ALK Q9UM73 1/20 0.38
KMT2A Q03164 1/20 0.38
METAP2 P50579 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434051 0.79 PDGFRB (0.52) PDGFRBAURKATTKAURKBINCENP
SCHEMBL7430163 0.78 CYP11B1 (0.47) PDGFRBAURKATTKAURKBINCENP
SCHEMBL9565370 0.78 PDGFRB (0.46) PDGFRBAURKATTKAURKBINCENP
SCHEMBL9565317 0.77 SMN1; SMN2 (0.49) CYP2A6CYP3A4CYP2C9CYP2B6CYP2C19
SCHEMBL9565313 0.77 PDGFRB (0.46) PDGFRBAURKATTKAURKBINCENP
SCHEMBL7495544 0.77 PDGFRB (0.48) PDGFRBAURKATTKAURKBINCENP
SCHEMBL7440831 0.74 CYP2A6 (0.44) CYP2A6MAPK1CYP3A4CYP2E1CYP2C9
SCHEMBL9963331 0.74 CYP2A6 (0.46) PDGFRBAURKATTKAURKBINCENP
SCHEMBL1435835 0.71 CYP2A6 (0.54) PDGFRBCYP2A6MAPK1CYP3A4ALDH1A1
SCHEMBL7430157 0.71 MAPK1 (0.42) CYP2A6MAPK1CYP3A4CYP2E1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278161-A Racemic mixtures HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
EP-0464572-A2 Aminoacid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed