SCHEMBL9565336

SCHEMBL9565336

CSCCCc1nc(-c2cccnc2)cnc1Cl

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 9/20 0.41
CYP3A4 P08684 5/20 0.41
CYP2C9 P11712 5/20 0.39
CYP2C19 P33261 5/20 0.39
CYP2E1 P05181 4/20 0.39
CYP2B6 P20813 4/20 0.39
CYP2D6 P10635 3/20 0.39
MAPK1 P28482 2/20 0.39
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
PTK2 Q05397 1/20 0.38
CYP19A1 P11511 4/20 0.36
DUSP10 Q9Y6W6 1/20 0.36
ATR Q13535 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7328164 0.84 CYP2A6 (0.45) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL9565345 0.81 MAPK1 (0.40) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL7440831 0.77 CYP2A6 (0.44) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL9565370 0.76 PDGFRB (0.46) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL7430012 0.75 CYP11B1 (0.50) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL9565316 0.74 CYP2A6 (0.43) CYP2A6CYP3A4MAPK1HSP90AA1HSP90AB1
SCHEMBL7424771 0.70 MAPK1 (0.48) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL20543722 0.69 CYP11B1 (0.61) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL7436678 0.68 CYP2A6 (0.43) CYP2A6CYP3A4CYP2C9CYP2C19CYP2E1
SCHEMBL7438980 0.68 MAPK1 (0.39) CYP3A4CYP2D6MAPK1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543245-A1 Renin inhibiting amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed