SCHEMBL9565522

SCHEMBL9565522

O=C(O)C(F)(COCc1ccccc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
KDM4E B2RXH2 1/20 0.51
POLB P06746 1/20 0.51
TSHR P16473 1/20 0.50
CES1 P23141 1/20 0.48
NPSR1 Q6W5P4 1/20 0.47
MAPK1 P28482 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PTPN2 P17706 1/20 0.42
PTPN1 P18031 1/20 0.42
PTPN6 P29350 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9116753 0.84 TSHR (0.48) ALDH1A1KDM4EPOLBTSHRCES1
Trifluoroacetic Acid SCHEMBL27579421 0.82 TSHR (0.62) ALDH1A1KDM4EPOLBTSHRCES1
SCHEMBL8839506 0.81 KDM4E (0.55) ALDH1A1KDM4EPOLBTSHRCES1
SCHEMBL3547434 0.81 KDM4E (0.55) ALDH1A1KDM4EPOLBTSHRMAPK1
SCHEMBL28943134 0.80 LMNA (0.48) ALDH1A1KDM4EPOLBTSHRCES1
SCHEMBL1691754 0.79 KDM4E (0.53) ALDH1A1KDM4EPOLBTSHRMAPK1
SCHEMBL8157722 0.78 ALDH1A1 (0.61) ALDH1A1KDM4EPOLBTSHRCES1
SCHEMBL31397663 0.78 KDM4E (0.51) ALDH1A1KDM4EPOLBTSHRMAPK1
SCHEMBL3545416 0.78 KDM4E (0.51) ALDH1A1KDM4EPOLBTSHRMAPK1
SCHEMBL8840022 0.77 KDM4E (0.51) ALDH1A1KDM4EPOLBTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107793381-A The preparation method of the methanol of 3 fluoro-oxetane 3 and its intermediate 上海睿智化学研究有限公司 2018-03-13 CN disclosed
EP-0554025-A2 Fluorinated cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1993-08-04 EP disclosed