SCHEMBL9567472

SCHEMBL9567472

CCOC(=O)c1cccc2c(=O)c(C)c(C=Cc3ccccc3)oc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
LMNA P02545 4/20 0.47
KDM4E B2RXH2 3/20 0.47
ADORA3 P0DMS8 2/20 0.47
CYP1A2 P05177 1/20 0.47
CHRM2 P08172 1/20 0.47
CYP3A4 P08684 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47
ACHE P22303 1/20 0.47
SLC6A2 P23975 1/20 0.47
PDE4A P27815 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
KCNH2 Q12809 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
MAPT P10636 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9567471 1.00 ALDH1A1 (0.47) ALDH1A1LMNAKDM4EADORA3CYP1A2
SCHEMBL8876470 0.86 CYSLTR1 (0.44) ALDH1A1LMNAKDM4EADORA3CYP1A2
SCHEMBL8876466 0.86 CYSLTR1 (0.44) ALDH1A1LMNAKDM4EADORA3CYP1A2
SCHEMBL8878647 0.79 ALDH1A1 (0.69) ALDH1A1LMNAKDM4EADORA3CYP1A2
SCHEMBL9161742 0.78 STING1 (0.58) KDM4EGLAMEN1KMT2ASMN1; SMN2
SCHEMBL9164869 0.78 MCL1 (0.43) ALDH1A1LMNAKDM4EADORA3CYP3A4
SCHEMBL9164874 0.78 MCL1 (0.43) ALDH1A1LMNAKDM4EADORA3CYP3A4
SCHEMBL8875460 0.77 ALDH1A1 (0.67) ALDH1A1LMNAKDM4EADORA3CYP1A2
SCHEMBL8876847 0.75 CLEC4M (0.47) ALDH1A1LMNAKDM4EADORA3CYP1A2
SCHEMBL11329873 0.75 TSHR (0.54) ALDH1A1KDM4ECYP1A2CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040434-C Heterobicyclic compounds RECORDATI CHEM PHARM (CH) 1998-10-28 CN disclosed
CN-1079738-A Heterobicyclic compounds RECORDATI CHEM PHARM (CH) 1993-12-22 CN disclosed
WO-1993017007-A1 HETEROBICYCLIC COMPOUNDS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.P.A. (IT) 1993-09-02 WO disclosed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP disclosed