SCHEMBL9568947

SCHEMBL9568947

COc1ccnc(-c2cccc(Cl)c2[S+](C)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.49
CCR5 P51681 1/20 0.49
CCR8 P51685 1/20 0.49
P2RX7 Q99572 5/20 0.43
CCR9 P51686 1/20 0.40
PIK3CA P42336 2/20 0.39
PIK3CB P42338 2/20 0.39
PIK3CG P48736 2/20 0.39
NFE2L2 Q16236 3/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
NOS2 P35228 1/20 0.36
PHGDH O43175 1/20 0.36
CLK4 Q9HAZ1 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
TSHR P16473 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568979 0.85 CCR1 (0.50) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL9568937 0.84 CCR1 (0.49) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL27927335 0.80 CCR1 (0.58) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL27909626 0.80 CCR1 (0.61) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL10333255 0.78 CCR1 (0.54) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL25714905 0.77 GRM5 (0.43) CCR1CCR5CCR8CYP1A2TSHR
SCHEMBL10333299 0.77 CCR1 (0.50) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL9540847 0.77 PDE10A (0.45) CCR1CCR5CCR8P2RX7NOS3
SCHEMBL9569056 0.76 CCR1 (0.51) CCR1CCR5CCR8P2RX7CCR9
SCHEMBL10333632 0.73 CCR1 (0.56) CCR1CCR5CCR8P2RX7CCR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1070400-A Benzoglyoxaline FISONS PLC (GB) 1993-03-31 CN disclosed
EP-0526033-A1 Benzimidazoles FISONS plc (GB) 1993-02-03 EP disclosed