SCHEMBL9540847

SCHEMBL9540847

COc1ccnc(-c2cccc(Cl)c2[S+]([O-])c2nc3ccccc3[nH]2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.45
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
NPC1 O15118 8/20 0.40
RAB9A P51151 8/20 0.40
SMN1; SMN2 Q16637 6/20 0.40
ALDH1A1 P00352 4/20 0.40
TP53 P04637 2/20 0.40
MAPT P10636 2/20 0.39
AMY1A P0DUB6 1/20 0.39
RUNX1 Q01196 1/20 0.38
CBFB Q13951 2/20 0.37
PKM P14618 2/20 0.37
KDM4E B2RXH2 3/20 0.37
GPR55 Q9Y2T6 1/20 0.37
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539618 0.89 PDE10A (0.46) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL9538681 0.88 PDE10A (0.45) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL10333779 0.87 PDE10A (0.48) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL10333523 0.82 PDE10A (0.43) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL10333478 0.82 PDE10A (0.48) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL10333408 0.80 PDE10A (0.40) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL10333269 0.80 PDE10A (0.44) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL6474693 0.78 PDE10A (0.43) PDE10ANOS3NOS1NOS2NPC1
SCHEMBL9568947 0.77 CCR1 (0.49) NOS3NOS1NOS2ALDH1A1CCR1
SCHEMBL10333166 0.77 PDE10A (0.40) PDE10ANOS3NOS1NOS2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993002077-A1 BENZIMIDAZOLES FISONS PLC (GB) 1993-02-04 WO claimed
EP-0526033-A1 Benzimidazoles FISONS plc (GB) 1993-02-03 EP claimed
EP-0526033-A1 Benzimidazoles FISONS plc (GB) 1993-02-03 EP disclosed