SCHEMBL9569776

SCHEMBL9569776

Cc1cc(NC(=O)NS(=O)(=O)c2ccc3[nH]ccc3c2)ccc1C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.55
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
EPHX1 P07099 2/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
MAOA P21397 2/20 0.42
MAOB P27338 1/20 0.42
NOTUM Q6P988 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9569790 0.88 IDH1 (0.48) IDH1HDAC3HDAC4HDAC1HDAC7
SCHEMBL9569774 0.78 ESR1 (0.52) MEN1KMT2AHDAC3HDAC4HDAC1
SCHEMBL22803273 0.74 IDH1 (0.53) IDH1HDAC3HDAC4HDAC1HDAC7
SCHEMBL9569788 0.74 ESR1 (0.62) MEN1KMT2AHDAC3HDAC4HDAC1
SCHEMBL22803696 0.71 NPC1 (0.67) EPHX1NPC1RAB9AMAOAMAOB
SCHEMBL22803968 0.71 ESR1 (0.62) IDH1EPHX1NPC1RAB9AMAOA
SCHEMBL15702552 0.71 IDH1 (1.00) IDH1
SCHEMBL22803271 0.70 EPHX1 (0.51) IDH1MEN1KMT2AEPHX1NPC1
SCHEMBL12175766 0.70 PKM (0.63) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL17664180 0.70 IDH1 (0.61) IDH1KMT2AEPHX1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560554-A2 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-09-15 EP disclosed
US-5169860-A Benzofuran or benzothiophene arylsulfonylureas ELI LILLY AND COMPANY (US) 1992-12-08 US disclosed