SCHEMBL9569790

SCHEMBL9569790

O=C(Nc1ccc(C(F)(F)F)c(Cl)c1)NS(=O)(=O)c1ccc2[nH]ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.48
MAOB P27338 4/20 0.46
MAOA P21397 2/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA7 P43166 2/20 0.45
CA9 Q16790 2/20 0.45
TRPV1 Q8NER1 2/20 0.45
EPHX1 P07099 2/20 0.43
KDR P35968 1/20 0.43
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
HDAC1 Q13547 2/20 0.42
BRAF P15056 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9569776 0.88 IDH1 (0.55) IDH1MAOBMAOAEPHX1NPC1
SCHEMBL9569774 0.82 ESR1 (0.52) MAOBMAOACA1CA2CA9
SCHEMBL9524746 0.81 CA2 (0.53) CA1CA2CA7CA9EPHX1
SCHEMBL22803870 0.79 ESR1 (0.57) IDH1MAOBMAOATRPV1KDR
SCHEMBL22803700 0.78 MAOB (0.54) IDH1MAOBMAOACA1CA2
SCHEMBL8761299 0.76 GFER (0.44) CA1CA2CA7CA9KDR
SCHEMBL9478768 0.75 CA2 (0.44) CA1CA2CA7CA9TRPV1
SCHEMBL9478180 0.75 CA2 (0.44) CA1CA2CA7CA9TRPV1
SCHEMBL22803273 0.74 IDH1 (0.53) IDH1MAOBMAOAEPHX1NPC1
SCHEMBL13675794 0.74 KDR (0.48) MAOBMAOACA9KDRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560554-A2 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-09-15 EP disclosed
US-5169860-A Benzofuran or benzothiophene arylsulfonylureas ELI LILLY AND COMPANY (US) 1992-12-08 US disclosed