SCHEMBL9575142

SCHEMBL9575142

Cc1c(Br)ccc2nc(N)nc(N)c12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.47
SLC2A1 P11166 1/20 0.47
DCPS Q96C86 1/20 0.45
KCNH2 Q12809 2/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ESR1 P03372 1/20 0.42
CHRM2 P08172 1/20 0.42
HTR1A P08908 1/20 0.42
MAPT P10636 1/20 0.42
CHRM1 P11229 1/20 0.42
HPGD P15428 1/20 0.42
MAOA P21397 1/20 0.42
DRD1 P21728 1/20 0.42
ACHE P22303 1/20 0.42
PTGS1 P23219 1/20 0.42
SLC6A2 P23975 1/20 0.42
PDE4A P27815 1/20 0.42
OPRM1 P35372 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8389989 0.81 DCPS (0.51) DHFRSLC2A1DCPSKCNH2MEN1
SCHEMBL4029524 0.81 DHFR (0.49) DHFRSLC2A1DCPSKCNH2MEN1
Hydrochloric Acid SCHEMBL6603234 0.79 DHFR (0.47) DHFRSLC2A1DCPSKCNH2MEN1
Hydrochloric Acid SCHEMBL27593037 0.79 DHFR (0.47) DHFRSLC2A1DCPSKCNH2MEN1
Hydrochloric Acid SCHEMBL6600020 0.79 DHFR (0.47) DHFRSLC2A1DCPSKCNH2MEN1
SCHEMBL25167004 0.78 DHFR (0.42) DHFRSLC2A1DCPSKCNH2
SCHEMBL30400707 0.78 DHFR (0.42) DHFRSLC2A1DCPSKCNH2
SCHEMBL8390658 0.78 SLC2A1 (0.49) DHFRSLC2A1KCNH2
SCHEMBL9575141 0.78 DHFR (0.46) DHFRSLC2A1DCPSKCNH2
SCHEMBL8036167 0.76 DHFR (0.45) DHFRSLC2A1DCPSKCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253396-B1 PROCESS FOR PREPARING 5,6-SUBSTITUTED-2,4-QUINAZOLINEDIAMINES AND INTERMEDIATES WARNER-LAMBERT COMPANY (US) 1993-03-17 EP claimed
EP-0253396-A2 Process for preparing 5,6-substituted-2,4-quinazolinediamines and intermediates WARNER-LAMBERT COMPANY (US) 1988-01-20 EP claimed
EP-0253396-B1 PROCESS FOR PREPARING 5,6-SUBSTITUTED-2,4-QUINAZOLINEDIAMINES AND INTERMEDIATES WARNER-LAMBERT COMPANY (US) 1993-03-17 EP disclosed
EP-0253396-A2 Process for preparing 5,6-substituted-2,4-quinazolinediamines and intermediates WARNER-LAMBERT COMPANY (US) 1988-01-20 EP disclosed
US-4677219-A Substituted benzonitriles WARNER-LAMBERT COMPANY (US) 1987-06-30 US disclosed