SCHEMBL9580689

SCHEMBL9580689

CCCCCCCCCOc1ccsc1C(=O)OC

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.70
MEN1 O00255 2/20 0.62
CYP1A2 P05177 1/20 0.62
MAPT P10636 3/20 0.48
ALDH1A1 P00352 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
SMPD1 P17405 4/20 0.45
LMNA P02545 2/20 0.44
NR1I2 O75469 1/20 0.44
CHRM2 P08172 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADRA2A P08913 1/20 0.44
OPRK1 P41145 1/20 0.44
HTR2B P41595 1/20 0.44
SLC6A3 Q01959 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PPARG P37231 1/20 0.44
PTPN2 P17706 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9667534 0.94 KMT2A (0.74) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL20505231 0.89 KMT2A (0.77) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL7263863 0.83 RAB9A (0.52) KMT2AMEN1CYP1A2ALDH1A1TDP1
SCHEMBL4331526 0.83 KMT2A (1.00) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL28272334 0.82 KMT2A (0.69) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL11717055 0.80 CYP3A4 (0.52) KMT2AMEN1MAPTALDH1A1TDP1
SCHEMBL2453740 0.78 KMT2A (0.64) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL18095045 0.77 KMT2A (1.00) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL8199735 0.77 KMT2A (0.62) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL11752210 0.77 PPARG (0.42) KMT2AMEN1MAPTLMNANR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5140147-A None JP disclosed
JP-H05140147-A NEW THIENYL-NONATETRAENOIC ACID DERIVATIVE F HOFFMANN LA ROCHE AG 1993-06-08 JP disclosed
EP-0510473-A1 Thienyl-nonatetraenoic acid derivatives with anti-rheumatic activity F. HOFFMANN-LA ROCHE AG (CH) 1992-10-28 EP disclosed