SCHEMBL9585261

SCHEMBL9585261

COc1ccccc1OCC1OCC(CBr)O1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
GLA P06280 1/20 0.51
ADRA2C P18825 1/20 0.48
DRD4 P21917 5/20 0.43
CHRNB4 P30926 2/20 0.42
CHRNA3 P32297 2/20 0.42
HTR1A P08908 8/20 0.41
ADRA1D P25100 8/20 0.41
ADRA1A P35348 8/20 0.41
ADRA1B P35368 8/20 0.41
TDP1 Q9NUW8 1/20 0.37
AGTR1 P30556 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9584987 0.89 ALDH1A1 (0.51) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL9584274 0.86 ALDH1A1 (0.51) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL9585096 0.86 ALDH1A1 (0.51) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL9711767 0.81 ALDH1A1 (0.46) ALDH1A1GLAADRA2CDRD4HTR1A
SCHEMBL9585387 0.81 ALDH1A1 (0.51) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL7282918 0.80 ALDH1A1 (0.71) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL3634571 0.80 ALDH1A1 (0.71) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL29769262 0.80 ALDH1A1 (0.71) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL93244 0.80 ALDH1A1 (0.71) ALDH1A1GLAADRA2CDRD4CHRNB4
SCHEMBL9586088 0.80 PKM (0.52) ALDH1A1GLADRD4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5212316-A Respiratory system disorders BOEHRINGER MANNHEIM ITALIA (IT) 1993-05-18 US disclosed
EP-0303227-B1 ETHERS AND THIOETHERS HAVING THERAPEUTICAL ACTIVITY, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-02-05 EP disclosed
US-4968706-A MUCOLYTIC, ANTITUSSIVE, BRONCHODILATOR, ANTIINFLAMMATORY BOEHRINGER MANNHEIN ITALIA, S.P.A. (IT) 1990-11-06 US disclosed
EP-0303227-A1 Ethers and thioethers having therapeutical activity, their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1989-02-15 EP disclosed