SCHEMBL9585709

SCHEMBL9585709

O=[N+]([O-])c1ccc2c(c1)C(O)C(Br)CCO2

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.42
HSP90AA1 P07900 1/20 0.42
RAB9A P51151 6/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
NPC1 O15118 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
MAPT P10636 4/20 0.40
LMNA P02545 3/20 0.40
MAPK1 P28482 2/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
BAZ1A Q9NRL2 1/20 0.38
HTT P42858 1/20 0.38
CHRNB4 P30926 6/20 0.37
CHRNA3 P32297 6/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
PLK1 P53350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9585706 1.00 HTR1A (0.42) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL9585715 1.00 HTR1A (0.42) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL10481283 0.84 HTR1A (0.42) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL10481308 0.78 HSP90AA1 (0.42) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL6350114 0.78 HSP90AA1 (0.47) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL13725104 0.77 HSP90AA1 (0.42) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL6341448 0.75 RAB9A (0.41) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL12211579 0.75 HSP90AA1 (0.40) HTR1AHSP90AA1RAB9AMEN1KMT2A
SCHEMBL8137807 0.75 CYP1A2 (0.43) HSP90AA1RAB9AMEN1KMT2ANPC1
SCHEMBL10407545 0.75 HSP90AA1 (0.38) HTR1AHSP90AA1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5194442-A 2,3,4,5-tetrahydro-1-benzoxepins, the use thereof and pharmaceutical products based on these compounds HOECHST AKTIENGESELLSCHAFT (DE) 1993-03-16 US disclosed
EP-0360131-A1 2,3,4,5-Tetrahydro-1-benzoxepines, method for their preparation, their use and pharmaceutical compositions based on these compounds HOECHST AKTIENGESELLSCHAFT (DE) 1990-03-28 EP disclosed