SCHEMBL9596048

SCHEMBL9596048

CS(=O)(=O)O[C@@H]1C[C@H](CC(CNC(=O)OCc2ccc([N+](=O)[O-])cc2)C(N)=O)N(C(=O)OCc2ccc([N+](=O)[O-])cc2)C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
ALDH1A1 P00352 2/20 0.35
TGM2 P21980 1/20 0.34
ABCB1 P08183 1/20 0.34
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.33
CTSL P07711 1/20 0.33
CCR5 P51681 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
BMP1 P13497 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9596622 0.86 DPP8 (0.40) DPP8DPP9ALDH1A1TGM2ABCB1
SCHEMBL8106429 0.83 DPP8 (0.36) DPP8DPP9ALDH1A1TGM2ABCB1
SCHEMBL7859861 0.83 PSEN1 (0.40) DPP8DPP9ALDH1A1MAPTHPGD
SCHEMBL8109280 0.83 DPP8 (0.40) DPP8DPP9ALDH1A1TGM2MAPT
SCHEMBL9595372 0.82 DPP8 (0.42) DPP8DPP9ALDH1A1TGM2ABCB1
SCHEMBL9137731 0.82 HTT (0.39) ALDH1A1MAPTHPGDTDP1
SCHEMBL7859716 0.82 PSEN1 (0.39) DPP8DPP9ALDH1A1MAPTRAB9A
SCHEMBL9519366 0.82 DPP8 (0.42) DPP8DPP9ALDH1A1TGM2ABCB1
SCHEMBL8098250 0.82 DPP8 (0.38) DPP8DPP9ALDH1A1TGM2ABCB1
SCHEMBL7805407 0.81 ALDH1A1 (0.41) ALDH1A1MAPTHPGDCCR5TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993011128-A1 AMINOALKYLPYRROLIDINYLTHIOCARBAPENEM DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-10 WO disclosed