SCHEMBL9601423

SCHEMBL9601423

CCOC(=O)CCCCON=C(c1cccnc1)c1cc(OC)c(OC)c(OC)c1

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 16/20 0.74
TBXA2R P21731 2/20 0.48
CYP1A1 P04798 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP1B1 Q16678 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9601416 1.00 TBXAS1 (0.74) TBXAS1TBXA2RCYP1A1CYP1A2CYP1B1
SCHEMBL10659433 0.89 TBXAS1 (0.93) TBXAS1TBXA2R
SCHEMBL9601906 0.88 TBXA2R (0.62) TBXAS1TBXA2R
SCHEMBL9601898 0.88 TBXA2R (0.62) TBXAS1TBXA2R
SCHEMBL9601366 0.84 TBXAS1 (0.85) TBXAS1TBXA2R
SCHEMBL9601354 0.84 TBXAS1 (0.85) TBXAS1TBXA2R
SCHEMBL9601778 0.82 TBXAS1 (0.70) TBXAS1TBXA2R
SCHEMBL9601773 0.82 TBXAS1 (0.70) TBXAS1TBXA2R
SCHEMBL9601397 0.78 TBXAS1 (0.74) TBXAS1TBXA2R
SCHEMBL9601393 0.78 TBXAS1 (0.74) TBXAS1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221601-B1 [[[(3-Pyridinyl)methylen]amino]oxy]alkanoic acids and esters JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-10 EP disclosed
US-5180832-A Chemical intermediate for thromboxane A2 inhibitor JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-19 US disclosed
US-4963573-A INHIBIT BIOSYNTHESIS OF THROMBOXANE A2 JANSSEN PHARMACEUTICA N.V. (BE) 1990-10-16 US disclosed
US-4746671-A THROMBOXANE SYNTHETASE INHIBITION JANSSEN PHARMACEUTICA N.V. (BE) 1988-05-24 US disclosed
EP-0221601-A1 [[[(3-Pyridinyl)methylen]amino]oxy]alkanoic acids and esters JANSSEN PHARMACEUTICA N.V. (BE) 1987-05-13 EP disclosed