SCHEMBL9601699

SCHEMBL9601699

O=C(NCCN1CCC(Nc2nc3cncnc3n2Cc2ccc(F)cc2)CC1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 4/20 0.52
KCNH2 Q12809 5/20 0.50
NR4A2 P43354 1/20 0.50
TP53 P04637 5/20 0.48
HRH1 P35367 2/20 0.47
HRH4 Q9H3N8 2/20 0.47
USP2 O75604 3/20 0.46
CYP1A2 P05177 3/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2C19 P33261 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TMEM97 Q5BJF2 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
CYP2D6 P10635 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
MLNR O43193 1/20 0.46
CACNA1F O60840 1/20 0.46
EED O75530 1/20 0.46
ABCB11 O95342 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9603207 0.89 KCNH2 (0.44) SSTR5KCNH2NR4A2TP53HRH1
SCHEMBL9564813 0.88 ALDH1A1 (0.47) SSTR5KCNH2NR4A2TP53HRH1
Fumaric Acid SCHEMBL9564986 0.87 SSTR5 (0.42) SSTR5KCNH2NR4A2TP53HRH1
Fumaric Acid SCHEMBL9565040 0.87 SSTR5 (0.46) SSTR5KCNH2NR4A2TP53HRH1
SCHEMBL9564777 0.86 KCNH2 (0.44) SSTR5KCNH2NR4A2TP53HRH1
SCHEMBL11471515 0.86 TP53 (0.61) SSTR5KCNH2NR4A2TP53TMEM97
SCHEMBL9602108 0.85 KCNH2 (0.49) SSTR5KCNH2NR4A2TP53HRH1
SCHEMBL9564822 0.85 KCNH2 (0.48) SSTR5KCNH2NR4A2TP53HRH1
SCHEMBL9565058 0.84 SSTR5 (0.54) SSTR5KCNH2NR4A2TP53HRH1
SCHEMBL9564985 0.83 SSTR5 (0.51) SSTR5KCNH2NR4A2TP53HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed