SCHEMBL9602886

SCHEMBL9602886

COc1ccc(CC2(N)N=CNC=C2N)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
CYP2D6 P10635 2/20 0.37
ALDH1A1 P00352 2/20 0.37
ATM Q13315 1/20 0.37
IDO1 P14902 3/20 0.37
AGXT P21549 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37
MMP2 P08253 3/20 0.36
MMP9 P14780 3/20 0.36
MMP8 P22894 3/20 0.36
MMP13 P45452 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
HPGD P15428 1/20 0.35
SLC6A4 P31645 1/20 0.35
AOC3 Q16853 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2388622 0.75 TDP1 (0.37) ALDH1A1CYP1A2CYP2C19MAPK1TDP1
SCHEMBL9602890 0.69 ALDH1A1 (0.37) LMNACYP2D6ALDH1A1ATMIDO1
SCHEMBL1824702 0.68 MAOB (0.55) CYP2D6ALDH1A1IDO1AGXTTAAR1
SCHEMBL30906675 0.67 DAO (0.33) LMNACYP2D6ALDH1A1ATMIDO1
Hydrochloric Acid SCHEMBL30293103 0.66 MAOB (0.53) ALDH1A1IDO1AGXTTAAR1SLC6A4
SCHEMBL30110627 0.66 ALDH1A1 (0.37) LMNACYP2D6ALDH1A1ATMIDO1
SCHEMBL31266473 0.65 POLB (0.35) LMNACYP2D6ALDH1A1ATMIDO1
SCHEMBL1822033 0.65 MAOB (0.47) IDO1AGXTTAAR1SLC6A4
SCHEMBL1824988 0.64 SLC6A4 (0.46) IDO1AGXTTAAR1SLC6A4
Hydrochloric Acid SCHEMBL3966019 0.64 IDO1 (0.47) IDO1AGXTTAAR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed