SCHEMBL9602890

SCHEMBL9602890

COc1ccc(CC2(N)NC=NC=C2N)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
CYP2D6 P10635 1/20 0.37
ATM Q13315 1/20 0.37
IDO1 P14902 3/20 0.37
AGXT P21549 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
MMP8 P22894 2/20 0.36
MMP13 P45452 2/20 0.36
LMNA P02545 2/20 0.35
HPGD P15428 1/20 0.35
SLC6A4 P31645 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAOB P27338 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602886 0.69 LMNA (0.38) ALDH1A1CYP2D6ATMIDO1AGXT
SCHEMBL1824702 0.68 MAOB (0.55) ALDH1A1CYP2D6IDO1AGXTTAAR1
SCHEMBL9602820 0.67 MGMT (0.34) ALDH1A1
SCHEMBL4456076 0.67 ALDH1A1 (0.38) ALDH1A1CYP2D6ATMIDO1AGXT
SCHEMBL1822033 0.65 MAOB (0.47) IDO1AGXTTAAR1SLC6A4MAOB
Hydrochloric Acid SCHEMBL3966019 0.64 IDO1 (0.47) IDO1AGXTTAAR1SLC6A4MAOB
SCHEMBL1824988 0.64 SLC6A4 (0.46) IDO1AGXTTAAR1SLC6A4MAOB
SCHEMBL4868046 0.64 TDP1 (0.52) ALDH1A1IDO1AGXTTAAR1SLC6A4
Hydrochloric Acid SCHEMBL3967323 0.63 IDO1 (0.46) IDO1AGXTTAAR1SLC6A4MAOB
SCHEMBL491284 0.62 IDO1 (0.42) ALDH1A1CYP2D6IDO1AGXTTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206415-B1 (4-PIPERIDINYLMETHYL AND -HETERO)PURINES JANSSEN PHARMACEUTICA N.V. (BE) 1993-01-27 EP disclosed