SCHEMBL9602995

SCHEMBL9602995

CC(C[O])Nc1ncccn1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
NPC1 O15118 2/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP2C19 P33261 1/20 0.36
MAPK1 P28482 1/20 0.36
FDPS P14324 1/20 0.35
KDM4E B2RXH2 2/20 0.33
FFAR2 O15552 1/20 0.33
MAPKAPK2 P49137 1/20 0.32
EDNRA P25101 1/20 0.32
ASPH Q12797 1/20 0.32
KDM8 Q8N371 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9272660 0.80 ALDH1A1 (0.48) ALDH1A1NPC1MEN1RAB9AKMT2A
SCHEMBL9602997 0.78 KCNH3 (0.43) ALDH1A1LMNAHTTNPC1MEN1
SCHEMBL30593321 0.77 TLR8 (0.48) ALDH1A1NPC1CYP2C19TSHR
SCHEMBL24567768 0.77 TLR8 (0.48) ALDH1A1NPC1CYP2C19TSHR
SCHEMBL146979 0.75 CYP2C19 (0.39) ALDH1A1LMNAHTTNPC1MEN1
Isaxonine SCHEMBL1270289 0.74 KCNH3 (0.43) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL10125355 0.70 CYP2C19 (0.39) ALDH1A1LMNAHTTNPC1MEN1
SCHEMBL13736558 0.70 IDH1 (0.41) ALDH1A1LMNAHTTCYP2C19FFAR2
SCHEMBL10154754 0.70 IDH1 (0.41) ALDH1A1LMNAHTTCYP2C19FFAR2
SCHEMBL1905978 0.70 CYP2C19 (0.39) ALDH1A1LMNAHTTNPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0232623-B1 1-CARBACEPHALOSPORIN ANTIBIOTICS ELI LILLY AND COMPANY (US) 1993-03-17 EP disclosed
US-4892942-A 1-CARBA (DETHIA)CEPHALOSPORINS ELI LILLY AND COMPANY (US) 1990-01-09 US disclosed
US-4791106-A 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1988-12-13 US disclosed
EP-0232623-A1 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1987-08-19 EP disclosed