SCHEMBL9604885

SCHEMBL9604885

O=C(OCC(OC(=O)c1ccccc1)c1nc2c(C(F)(F)F)cccc2c(O)c1C(=O)Nc1nccs1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SCD O00767 1/20 0.38
KCNK3 O14649 1/20 0.37
KCNK9 Q9NPC2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837932 0.92 NPC1 (0.42) NPC1RAB9AHPGDSMN1; SMN2SCD
SCHEMBL9605133 0.88 RAB9A (0.38) NPC1RAB9AHPGDSMN1; SMN2MEN1
SCHEMBL9602628 0.86 RAB9A (0.39) NPC1RAB9AHPGDSMN1; SMN2MEN1
SCHEMBL9605284 0.83 RAB9A (0.39) NPC1RAB9AHPGDSMN1; SMN2MEN1
SCHEMBL9837751 0.83 NPC1 (0.41) NPC1RAB9AHPGDSMN1; SMN2MEN1
SCHEMBL9838903 0.82 RAB9A (0.40) NPC1RAB9AHPGDSMN1; SMN2MEN1
SCHEMBL10667122 0.81 KDM4E (0.40) MEN1KMT2A
SCHEMBL10518993 0.81 NPC1 (0.40) NPC1RAB9AHPGDSMN1; SMN2LMNA
SCHEMBL9839261 0.81 NPC1 (0.40) NPC1RAB9AHPGDSMN1; SMN2MEN1
SCHEMBL11620300 0.81 HTT (0.44) NPC1RAB9AHPGDSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214004-B1 4-OH-QUINOLINE-CARBOXYLIC-ACID DERIVATIVES SUBSTITUTED IN POSITION 2 BY A DIHYDROXY-SUBSTITUTED GROUP, POSSIBLY ETHERIFIED OR ESTERIFIED, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-03-31 EP disclosed
US-4988708-A 3-Carbamoyl-4-hydroxy-2-carboxylmethyl quinoline analgesics, antiinflammatory agents ROUSSEL UCLAF (FR) 1991-01-29 US disclosed
US-4845105-A 4-OH-quinoline carboxylic acid amides having analgesic and anti-inflammatory activity ROUSSEL UCLAF (FR) 1989-07-04 US disclosed