SCHEMBL9607091

SCHEMBL9607091

CCOC(=O)/C=C(\Nc1ccccc1)c1ccc(Cc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.45
PPARG P37231 2/20 0.45
PPARA Q07869 2/20 0.45
POLB P06746 2/20 0.44
CTNNB1 P35222 1/20 0.44
TCF7L2 Q9NQB0 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
PDK1 Q15118 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK3 Q15120 1/20 0.42
PDK4 Q16654 1/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
FAAH O00519 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
THRB P10828 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
FPR2 P25090 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9607506 1.00 EPHX2 (0.45) EPHX2PPARGPPARAPOLBCTNNB1
SCHEMBL8515651 0.87 KMT2A (0.48) EPHX2CTNNB1TCF7L2SMN1; SMN2CYP1A2
SCHEMBL9607492 0.86 POLB (0.43) EPHX2PPARGPPARAPOLBSMN1; SMN2
SCHEMBL8535567 0.86 SMN1; SMN2 (0.49) POLBSMN1; SMN2ALDH1A1CYP1A2CYP2C19
SCHEMBL8535569 0.86 SMN1; SMN2 (0.49) POLBSMN1; SMN2ALDH1A1CYP1A2CYP2C19
SCHEMBL9607414 0.85 TRPV1 (0.47) EPHX2PPARGPPARAPOLBSMN1; SMN2
SCHEMBL9607177 0.83 KMT2A (0.50) EPHX2POLBSMN1; SMN2ALDH1A1MAPT
SCHEMBL9607090 0.83 PDE2A (0.42) EPHX2PPARGPPARAPOLBSMN1; SMN2
SCHEMBL9607491 0.82 HTR1D (0.43) EPHX2SMN1; SMN2ALDH1A1MAPTLMNA
SCHEMBL3858960 0.80 GAA (0.51) SMN1; SMN2ALDH1A1MAPTLMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed