SCHEMBL9607432

SCHEMBL9607432

CCCc1nc(N)nc(C)c1CC(C)C

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 11/20 0.41
TLR7 Q9NYK1 8/20 0.41
HSP90AA1 P07900 1/20 0.37
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HEXA P06865 1/20 0.36
HEXB P07686 1/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15434720 0.86 TLR8 (0.39) TLR8TLR7MAPK1KDM4EHEXA
SCHEMBL9286489 0.81 NOS3 (0.39) TLR8TLR7MAPK1KDM4EALDH1A1
SCHEMBL9286486 0.79 TLR8 (0.52) TLR8TLR7
SCHEMBL15434700 0.74 TLR8 (0.45) TLR8TLR7HSP90AA1MAPK1HEXA
SCHEMBL15429559 0.74 MAPK1 (0.34) TLR8TLR7MAPK1KDM4EALDH1A1
SCHEMBL16229363 0.73 TLR8 (0.65) TLR8TLR7
SCHEMBL17229299 0.70 NOS2 (0.44) KDM4EALDH1A1
SCHEMBL27544017 0.70 HEXA (0.49) MAPK1KDM4EHEXAHEXBPOLB
SCHEMBL2072604 0.68 HEXA (0.46) HSP90AA1MAPK1KDM4EHEXAHEXB
SCHEMBL15429545 0.68 TLR8 (0.42) TLR8TLR7MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071519-A1 BENZOXAZEPINES AS INHIBITORS OF P13K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed