SCHEMBL9607519

SCHEMBL9607519

CN(C)Cc1ncc(CC(F)(F)F)cn1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
HRH3 Q9Y5N1 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16459436 0.75 SLC6A2 (0.31)
SCHEMBL16479755 0.75
SCHEMBL24655826 0.74 CHRNB2 (0.33) CHRNB2CHRNA4HRH3ALDH1A1TSHR
SCHEMBL16476944 0.73 CYP2C19 (0.33)
SCHEMBL25680871 0.72 ALOX15 (0.38) CHRNB2CHRNA4HRH3ALDH1A1TSHR
SCHEMBL22719101 0.71 TRPV1 (0.36) CHRNB2CHRNA4
SCHEMBL12092560 0.70 POLB (0.41) CHRNB2CHRNA4
SCHEMBL21789415 0.68 CYP2C19 (0.48) CHRNB2CHRNA4HRH3ALDH1A1TSHR
SCHEMBL12828104 0.68 CYP2A6 (0.33)
SCHEMBL16476787 0.66 CYP2C19 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071519-A1 BENZOXAZEPINES AS INHIBITORS OF P13K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed