SCHEMBL960971

SCHEMBL960971

CN(C)CC(C)(C)COc1ccc2[nH]c(-c3cc(NC(=O)c4cnn(Cc5ccc(Cl)s5)c4)c[nH]c3=O)cc2c1

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.32
PLA2G1B P04054 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ATG4B Q9Y4P1 1/20 0.31
TAS2R8 Q9NYW2 1/20 0.31
RAF1 P04049 2/20 0.31
BRAF P15056 2/20 0.31
ALDH1A1 P00352 1/20 0.31
KDR P35968 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL950079 0.89 ALDH1A1 (0.41) KLKB1ALDH1A1KDR
SCHEMBL31060778 0.89 ALDH1A1 (0.41) KLKB1ALDH1A1KDR
SCHEMBL950040 0.89 KLKB1 (0.36) KLKB1PLA2G1BCYP1A2CYP3A4CYP2D6
SCHEMBL12945028 0.86
SCHEMBL950481 0.83 ALDH1A1 (0.42) KLKB1PLA2G1BCYP1A2CYP3A4CYP2D6
SCHEMBL964521 0.82 ITK (0.36) MAPTTAS2R8KDR
SCHEMBL949097 0.81 RPS6KA2 (0.40) KLKB1ALDH1A1
SCHEMBL15520154 0.80 KDR (0.35) MAPTSMN1; SMN2ALDH1A1KDR
SCHEMBL1002318 0.79 CHEK1 (0.47)
SCHEMBL951282 0.79 ALDH1A1 (0.40) KLKB1ALDH1A1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011010083-A1 INDOLYL-PYRIDONE DERIVATIVES VERNALIS (R & D) LTD (GB) 2011-01-27 WO claimed
WO-2011010083-A1 INDOLYL-PYRIDONE DERIVATIVES VERNALIS (R & D) LTD (GB) 2011-01-27 WO disclosed
WO-2011010083-A1 INDOLYL-PYRIDONE DERIVATIVES VERNALIS (R & D) LTD (GB) 2011-01-27 WO disclosed