SCHEMBL964521

SCHEMBL964521

O=C(Nc1c[nH]c(=O)c(-c2cc3ccccc3[nH]2)c1)c1cnn(Cc2ccc(Cl)s2)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.36
SCD5 Q86SK9 3/20 0.36
RPS6KA3 P51812 3/20 0.36
RPS6KA2 Q15349 2/20 0.36
RPS6KA1 Q15418 2/20 0.36
RPS6KA6 Q9UK32 2/20 0.36
PRSS12 P56730 1/20 0.35
CHEK1 O14757 1/20 0.34
KDR P35968 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
ROCK1 Q13464 4/20 0.34
STK33 Q9BYT3 1/20 0.34
TAS2R8 Q9NYW2 1/20 0.34
SCD O00767 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL947957 0.88 RPS6KA2 (0.46) ITKSCD5RPS6KA3RPS6KA2RPS6KA1
SCHEMBL951873 0.87 KMT2A (0.44) ITKSCD5RPS6KA3RPS6KA2RPS6KA1
SCHEMBL1002318 0.86 CHEK1 (0.47) CHEK1
SCHEMBL948561 0.85 ITK (0.50) ITKSCD5RPS6KA3RPS6KA2RPS6KA1
SCHEMBL948091 0.85 ALDH1A1 (0.41) SCD5RPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL950898 0.85 KLKB1 (0.45) ITKRPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL951550 0.83 KMT2A (0.40) ITKRPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL949397 0.83 KLKB1 (0.39) ITKRPS6KA3RPS6KA2RPS6KA1RPS6KA6
SCHEMBL960971 0.82 KLKB1 (0.32) KDRMAPTTAS2R8
SCHEMBL949207 0.82 SCD (0.44) SCD5SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011010083-A1 INDOLYL-PYRIDONE DERIVATIVES VERNALIS (R & D) LTD (GB) 2011-01-27 WO disclosed
WO-2011010083-A1 INDOLYL-PYRIDONE DERIVATIVES VERNALIS (R & D) LTD (GB) 2011-01-27 WO disclosed