SCHEMBL9622945

SCHEMBL9622945

CNc1ncc(C(N)=O)c(OC)n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.44
NNMT P40261 3/20 0.44
GSK3B P49841 1/20 0.44
LRRK2 Q5S007 1/20 0.43
MAPK3 P27361 1/20 0.42
SYK P43405 5/20 0.42
LCK P06239 3/20 0.41
MAPK8 P45983 3/20 0.41
MAPK9 P45984 2/20 0.41
MAPK14 Q16539 2/20 0.41
KDR P35968 1/20 0.41
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10827865 0.85 POLB (0.47) GSK3BLRRK2LCKMAPK14KDR
SCHEMBL15946663 0.84 LCK (0.46) LRRK2LCKMAPK14KDR
SCHEMBL14590441 0.79 RAB9A (0.48)
SCHEMBL23775486 0.78 NNMT (0.51) NNMTSYK
SCHEMBL762022 0.78 SYK (0.52) NNMTLRRK2SYKMAPK8MAPK9
SCHEMBL3192298 0.78 NNMT (0.47) NNMTGSK3BSYKMAPK8
SCHEMBL30962568 0.77 NNMT (0.46) NNMTGSK3BLRRK2SYK
SCHEMBL30962899 0.76 JAK3 (0.58) GSK3BSYKKDR
SCHEMBL25224808 0.74 NNMT (0.44) NNMTGSK3B
SCHEMBL5765616 0.74 POLB (0.49) NNMTLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5137895-A Antiemetic, anxiolytic, gastric emptying and serotonin modulating activity A. H. ROBINS COMPANY, INCORPORATED (US) 1992-08-11 US disclosed